Phase 5l selection gate — K1141 fragment ladder

Evaluates 4 fragment lengths × 2 variants on AF3 server outputs vs Phase 5d snap_010 (full-length E1659A MD-relaxed). Gate: pocket-pLDDT ≥ 80, K1141-ring Cα RMSD < 1.5 Å, whole-fragment Cα RMSD < 2.5 Å.

Fragment (aa)Variantpocket pLDDTring pLDDTfrag RMSD (Å)ring RMSD (Å)pTMrank-scoreVerdict
121wt81.581.18.505.850.510.60❌ FAIL
121e1659a84.183.78.223.350.600.69❌ FAIL
151wt78.078.25.381.940.640.71❌ FAIL
151e1659a78.778.74.870.970.650.73❌ FAIL
181wt80.880.66.572.650.670.73❌ FAIL
181e1659a79.178.86.082.480.650.71❌ FAIL
221wt81.781.75.231.320.730.81❌ FAIL
221e1659a81.681.55.551.400.730.81❌ FAIL

No fragment passes the strict gate.