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Hypotheses
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H01 · Pharmacochaperone E1659A
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artifacts
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phase8h_lite
Folder: hypotheses/h01-pharmacochaperone/artifacts/phase8h_lite
10 items under this folder.
Apr 26, 2026
result_09_pbpk_dose_sweep
Apr 26, 2026
Phase 8h-lite · Light computational evidence package for H01
strc
h01
summary
paper-ready
Apr 26, 2026
Phase 8h-lite #1 · K1141 pocket druggability profile
strc
h01
pocket
druggability
sitemap
Apr 26, 2026
Phase 8h-lite #2 · RWM permeability prediction for lead candidate
strc
h01
pkpd
round-window
permeability
salt-ma
Apr 26, 2026
Phase 8h-lite #3 · Off-target selectivity charge proxy (inconclusive light)
strc
h01
off-target
selectivity
electrostatics
Apr 26, 2026
Phase 8h-lite #4 · Lead-pose ensemble stability vs K1141 across Phase 5d
strc
h01
ensemble
pose-stability
k1141
Apr 26, 2026
Phase 8h-lite #5 · Tanimoto vs known cochlear ototoxins
strc
h01
medchem
ototoxicity
tanimoto
Apr 26, 2026
Phase 8h-lite #6 · Tier-1 RWM permeability + Tanimoto refresh after Phase 7I lead pivot
strc
h01
tier1
rwm
tanimoto
prodrug
lead-pivot
Apr 26, 2026
Phase 8h-lite #7 · Cochlear-compartment PBPK ODE
strc
h01
pkpd
pbpk
intratympanic
cochlear-compartment
elx-02-lesson
Apr 26, 2026
Phase 8h-lite #8 · K1141 pocket vs stereocilin-partner interface map
strc
h01
structure
interface-map
allosteric
partner-binding
e1659a-domain